Preferred Label : protein kinase inhibitors;

MeSH definition : Agents that inhibit PROTEIN KINASES.;

MeSH synonym : inhibitors, protein kinase; kinase inhibitors, protein; Protein Kinase Inhibitor; Inhibitor, Protein Kinase; Kinase Inhibitor, Protein;

Is substance : O;

action pharmacologique : O;

Details


Main resources

You can consult :

Agents that inhibit PROTEIN KINASES.

https://pharmactuel.com/index.php/pharmactuel/article/view/1265
2019
false
false
false
false
France
comparative effectiveness research
treatment outcome
EGFR Gene Mutation
protein kinase inhibitors
protein-tyrosine kinases
antineoplastic agents
Gefitinib
Afatinib
clinical trials, phase iii as topic
antineoplastic agents
protein kinase inhibitors
lung neoplasms
lung neoplasms
carcinoma, non-small-cell lung
osimertinib
osimertinib
Tyrosine Kinase Inhibitors
critical appraisal or critical reading
carcinoma, non-small-cell lung
piperazines
piperazines
acrylamides
aniline compounds
acrylamides
aniline compounds

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Summary Safety Review - Vascular endothelial growth factor receptor tyrosine kinase inhibitors
https://hpr-rps.hres.ca/reg-content/resume-examen-innocuite-detail.php?lang=fr&linkID=SSR00213
2018
false
false
false
Canada
French
English
receptors, vascular endothelial growth factor
protein kinase inhibitors
soft tissue neoplasms
kidney neoplasms
liver neoplasms
arteries
aneurysm
Aortic Dissection
aorta
pazopanib
ponatinib
regorafenib
vandetanib
lenvatinib
administration, oral
risk assessment
pharmacovigilance note
Tyrosine Kinase Inhibitors
indoles
pyrroles
phenylurea compounds
niacinamide
niacinamide
imidazoles
indazoles
pyrimidines
sulfonamides
pyridazines
pyridines
piperidines
quinazolines
quinolines
Sorafenib
Sunitinib
Axitinib

---
http://www.sfendocrino.org/_images/mediatheque/articles/pdf/recommandations/2018_Immunotherapies%20/mced_94_bd.pdf
2018
false
false
false
France
French
immunotherapy
antibodies, monoclonal
consensus
continuity of patient care
Tyrosine Kinase Inhibitor
protein-tyrosine kinases
protein kinase inhibitors
TOR Serine-Threonine kinases
adrenal glands
pituitary gland
metabolism
endocrine system diseases
diabetes mellitus
Hypophysitis
hypothyroidism
adrenal insufficiency
Hormone Measurement
hormones
Tyrosine Kinase Inhibitors

---
https://pharmacomedicale.org/medicaments/par-specialites/item/inhibiteurs-de-proteines-kinases
2016
false
false
false
France
French
protein kinase inhibitors
drug information
protein kinase inhibitors
protein kinase

---
http://www.e-cancer.fr/Expertises-et-publications/Catalogue-des-publications/Medicaments-ciblant-BCR-ABL-Imatinib-Dasatinib-Nilotinib-Bosutinib-Ponatinib-Medicament-ciblant-JAK-Ruxolitinib-Anticancereux-par-voie-orale-informer-prevenir-et-gerer-leurs-effets-indesirables
2016
false
false
false
France
French
practice guideline
antineoplastic agents
administration, oral
Drug-Related side effects and adverse reactions
Drug-Related side effects and adverse reactions
information dissemination
patient education as topic
drug interactions
Dasatinib
Imatinib Mesylate
fusion proteins, bcr-abl
protein kinase inhibitors
dasatinib
imatinib
nilotinib
nilotinib
bosutinib
ponatinib
ruxolitinib
janus kinases
ponatinib
ruxolitinib
bosutinib
continuity of patient care
pregnancy
Tyrosine Kinase Inhibitors
nilotinib
ruxolitinib
aniline compounds
nitriles
quinolines
imidazoles
pyridazines
pyrimidines
pyrazoles

---
http://www.e-cancer.fr/Expertises-et-publications/Catalogue-des-publications/Medicaments-ciblant-ALK-crizotinib-ceritinib
2016
false
false
false
France
French
guidelines for drug use
protein kinase inhibitors
crizotinib
carcinoma, non-small-cell lung
ceritinib
ceritinib
receptor Protein-Tyrosine kinases
antineoplastic agents
administration, oral
protein kinase inhibitors
ceritinib
Drug-Related side effects and adverse reactions
continuity of patient care
drug interactions
interdisciplinary communication
risk factors
drug monitoring
ceritinib
carcinoma, non-small-cell lung
ALK gene rearrangement positive
ALK protein, human
patients guideline
practice guideline
Tyrosine Kinase Inhibitors
pyrimidines
sulfones
pyrimidines
sulfones
pyrimidines
sulfones
receptor Protein-Tyrosine kinases
Crizotinib
Crizotinib
Crizotinib
Anaplastic Lymphoma Kinase

---
http://www.sciencedirect.com/science/article/pii/S0007455116000606
10.1016/j.bulcan.2016.02.001
2016
false
false
false
France
French
pregnancy
Tyrosine Kinase Inhibitor
protein kinase inhibitors
protein-tyrosine kinases
journal article
risk assessment
review of literature
fetus
abortion, spontaneous
abnormalities, drug-induced
antineoplastic agents
Tyrosine Kinase Inhibitors

---
http://www.e-cancer.fr/Expertises-et-publications/Catalogue-des-publications/Medicaments-ciblant-BRAF-en-monotherapie-vemurafenib-dabrafenib-Medicaments-ciblant-BRAF-ou-MEK-en-association-vemurafenib-cobimetinib-dabrafenib-trametinib
2016
false
false
false
France
French
guidelines for drug use
practice guideline
patients guideline
protein kinase inhibitors
protein kinase inhibitors
Drug-Related side effects and adverse reactions
administration, oral
drug interactions
vemurafenib
vemurafenib
antineoplastic combined chemotherapy protocols
vemurafenib
dabrafenib
dabrafenib
dabrafenib
BRAF protein, human
Metastatic Melanoma
melanoma
melanoma
neoplasm metastasis
BRAF Gene Mutation
continuity of patient care
drug monitoring
interdisciplinary communication
protein kinase inhibitors
vemurafenib
dabrafenib
pregnancy
imidazoles
oximes
imidazoles
oximes
proto-oncogene proteins b-raf
imidazoles
oximes
indoles
sulfonamides
indoles
sulfonamides
indoles
sulfonamides
Vemurafenib
Vemurafenib
Vemurafenib

---
BCR-ABL Tyrosine Kinase Inhibitors [GLEEVEC (imatinib mesylate), TASIGNA (nilotinib), BOSULIF (bosutinib), SPRYCEL (dasatinib), ICLUSIG (ponatinib hydrochloride)] - Risk of Hepatitis B Reactivation
http://canadiensensante.gc.ca/recall-alert-rappel-avis/hc-sc/2016/58222a-fra.php
2016
false
false
false
Canada
French
English
pharmacovigilance note
fusion proteins, bcr-abl
protein kinase inhibitors
Imatinib Mesylate
risk
hepatitis b virus
imatinib
nilotinib
nilotinib
bosutinib
bosutinib
Dasatinib
dasatinib
ponatinib hydrochloride
ponatinib
Tyrosine Kinase Inhibitor
Hepatitis B reactivation
guidelines for drug use
continuity of patient care
mass screening
hepatitis B
hepatitis B
Tyrosine Kinase Inhibitors
nilotinib
ponatinib
pyrimidines
imidazoles
pyridazines
aniline compounds
nitriles
quinolines

---
Summary Safety Review - Bcr-Abl Tyrosine Kinase Inhibitors - Assessing the Potential Harm to the Fetus
http://www.hc-sc.gc.ca/dhp-mps/medeff/reviews-examens/tki-ikt-fra.php
2016
false
false
false
Canada
French
English
pregnancy
fusion proteins, bcr-abl
protein kinase inhibitors
protein-tyrosine kinases
drug evaluation
risk assessment
fetus
contraception
abnormalities, drug-induced
Tyrosine Kinase Inhibitor
abortion, spontaneous
hematologic diseases
antineoplastic agents
administration, oral
pharmacovigilance
Tyrosine Kinase Inhibitors

---
https://www.jle.com/fr/revues/ito/e-docs/suivi_therapeutique_pharmacologique_des_inhibiteurs_de_proteines_kinases_305645/article.phtml
2015
false
false
false
France
French
journal article
protein kinase inhibitors
drug monitoring
dose-response relationship, drug
Precision Medicine
pharmacogenetics
protein kinase inhibitors
antineoplastic agents
antineoplastic agents
imatinib
protein-tyrosine kinases
enzyme inhibitors
enzyme inhibitors
continuity of patient care
Imatinib mesylate:MCnc:Pt:Ser/Plas:Qn:
chemistry techniques, analytical
protein kinase inhibitors
enzyme inhibitors
antineoplastic agents
Imatinib Mesylate
Imatinib Mesylate
Imatinib Mesylate
Tyrosine Kinase Inhibitors

---
http://www.pharmactuel.com/index.php/pharmactuel/article/view/942
2014
false
Canada
French
lung neoplasms
carcinoma, non-small-cell lung
journal article
lung neoplasms
carcinoma, non-small-cell lung
lung neoplasms
carcinoma, non-small-cell lung
antineoplastic agents
antibodies, monoclonal, humanized
angiogenesis inhibitors
protein kinase inhibitors
pyrazoles
pyridines
Erlotinib Hydrochloride
Pemetrexed
Bevacizumab
Gefitinib
Crizotinib

---
https://www.revmed.ch/RMS/2014/RMS-N-414/Rhumatologie-Une-nouvelle-option-therapeutique-dans-la-prise-en-charge-de-l-inflammation-chronique-en-rhumatologie-les-inhibiteurs-des-Janus-kinases
2014
false
false
false
Switzerland
piperidines
journal article
tofacitinib
protein kinase inhibitors
pyrimidines
pyrroles
tofacitinib
protein kinase inhibitors
piperidines
pyrimidines
pyrroles
arthritis, rheumatoid

---
https://www.ema.europa.eu/medicines/human/EPAR/Nexavar
2012
false
United Kingdom
English
French
phenylurea compounds
phenylurea compounds
niacinamide
syndication feed
treatment outcome
drug evaluation
orphan drug production
carcinoma, renal cell
pyridines
benzenesulfonates
antineoplastic agents
protein kinase inhibitors
sorafenib
pyridines
benzenesulfonates
antineoplastic agents
protein kinase inhibitors
sorafenib tosylate
sorafenib tosylate
drug evaluation
summary of product characteristics
package leaflet
Sorafenib
Sorafenib

---
http://www.has-sante.fr/portail/jcms/c_946059/torisel-temsirolimus-inhibiteur-de-proteine-kinase
http://www.has-sante.fr/portail/upload/docs/application/pdf/2010-03/torisel_-_ct-7303.pdf
2010
false
France
French
sirolimus
infusions, intravenous
orphan drug production
antineoplastic agents
carcinoma, renal cell
lymphoma, mantle-cell
temsirolimus
neoplasm recurrence, local
adult
aged
treatment outcome
temsirolimus
antineoplastic agents
protein kinase inhibitors
temsirolimus
protein kinase inhibitors
evaluation of the transparency committee
guidelines for drug use

---
https://www.jle.com/fr/revues/medecine/hma/e-docs/00/04/3A/C9/resume.md
2008
false
France
French
Imatinib Mesylate
protein kinase inhibitors
antineoplastic agents
dendritic cells
t-lymphocytes
killer cells, natural
leukemia, myelogenous, chronic, bcr-abl positive
journal article

---
http://www.omedit-centre.fr/portail/gallery_files/site/136/2953/5062/5139.pdf
2007
false
France
French
Erlotinib Hydrochloride
Cetuximab
drug eruptions
skin diseases
skin diseases
antineoplastic agents
protein kinase inhibitors
drug eruptions
practice guideline

---
http://www.msss.gouv.qc.ca/sujets/organisation/lutte-contre-le-cancer/documents/guides-cepo-pdf/CEPO-Tarceva_et_poumon_(2005-06).pdf
2005
false
false
Canada
French
English
Erlotinib Hydrochloride
protein kinase inhibitors
lung neoplasms
carcinoma, non-small-cell lung
lung neoplasms
carcinoma, non-small-cell lung
survival rate
lung neoplasms
carcinoma, non-small-cell lung
bibliography of medicine
Evidence-Based medicine
quebec
Tyrosine Kinase Inhibitors
erlotinib
graph
guidelines for drug use
ErbB Receptors

---
http://www.msss.gouv.qc.ca/sujets/organisation/lutte-contre-le-cancer/documents/guides-cepo-pdf/guide_utilisation_imatinib_2004.pdf
2004
false
false
Canada
French
English
Imatinib Mesylate
Imatinib Mesylate
Imatinib Mesylate
protein kinase inhibitors
Evidence-Based medicine
leukemia, myelogenous, chronic, bcr-abl positive
incidence
bibliography of medicine
antineoplastic agents
protein kinase inhibitors
antineoplastic agents
protein kinase inhibitors
survival rate
quebec
leukemia, myelogenous, chronic, bcr-abl positive
antineoplastic agents
imatinib
guidelines for drug use
graph

---
http://www.msss.gouv.qc.ca/sujets/organisation/lutte-contre-le-cancer/documents/guides-cepo-pdf/guide_utilisation_imatinib_2002.pdf
2002
false
false
Canada
French
Imatinib Mesylate
Imatinib Mesylate
antineoplastic agents
protein kinase inhibitors
gastrointestinal stromal tumors
gastrointestinal stromal tumors
incidence
bibliography of medicine
antineoplastic agents
protein kinase inhibitors
drug interactions
quebec
imatinib
guidelines for drug use

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06/06/2024


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