Preferred Label : lenvatinib;

MeSH note : a protein kinase inhibitor; structure in first source;

CISMeF synonym : E 7080; E7080 cpd;

MeSH synonym : 4-(3-chloro-4-(N'-cyclopropylureido)phenoxy)-7-methoxyquinoline-6-carboxamide; 4-(3-chloro-4-((cyclopropylaminocarbonyl)amino)phenoxy)-7-methoxy-6-quinolinecarboxamide;

MeSH hyponym : E-7080; E7080 mesylate; N-(4-((6-carbamoyl-7-methoxyquinolin-4-yl)oxy)-2-chlorophenyl)-N'-cyclopropylurea monomethanesulfonate; lenvatinib mesilate; lenvatinib methanesulfonate; Lenvima; E-7080 mesylate; ER-203492-00; E7080; 4-(3-chloro-4-(((cyclopropylamino)carbonyl)amino)phenoxy)-7-hydroxy-6-quinolinecarboxamide;

Related MeSH term : E7080 mesylate;

MeSH Related Number : 269N24780P; 3J78384F61;

Is substance : O;

UNII : EE083865G2;

InChIKey : WOSKHXYHFSIKNG-UHFFFAOYSA-N;

Details


Main resources

You can consult :


https://www.has-sante.fr/jcms/p_3420695/fr/lenvima-lenvatinib-cancer-de-l-endometre
2023
false
false
false
France
antineoplastic agents
protein kinase inhibitors
lenvatinib
antineoplastic combined chemotherapy protocols
pembrolizumab
Lenvatinib/Pembrolizumab Regimen
adult
Advanced Endometrial Carcinoma
Recurrent Endometrial Carcinoma
Refractory Endometrial Carcinoma
Unresectable Endometrial Carcinoma
administration, oral
evaluation of the transparency committee
lenvatinib
endometrial neoplasms

---
https://www.has-sante.fr/jcms/p_3334582/fr/lenvima-lenvatinib-carcinome-endometrial
2022
false
false
false
France
French
evaluation of the transparency committee
antineoplastic combined chemotherapy protocols
treatment outcome
insurance, health, reimbursement
Lenvatinib/Pembrolizumab Regimen
adult
Refractory Endometrial Carcinoma
Recurrent Endometrial Carcinoma
Advanced Endometrial Carcinoma
administration, oral
lenvatinib
antineoplastic agents
protein kinase inhibitors
lenvatinib
endometrial neoplasms

---
https://www.has-sante.fr/jcms/p_3324073/fr/kisplyx-lenvatinib
2022
false
false
false
France
treatment outcome
insurance, health, reimbursement
lenvatinib
administration, oral
lenvatinib
protein kinase inhibitors
protein kinase inhibitors
antineoplastic agents
antineoplastic agents
antineoplastic combined chemotherapy protocols
Lenvatinib/Pembrolizumab Regimen
pembrolizumab
clear cell renal cell carcinoma
Advanced Clear Cell Renal Cell Carcinoma
evaluation of the transparency committee
lenvatinib

---
https://www.has-sante.fr/jcms/p_3325606/fr/lenvima-lenvatinib
https://www.has-sante.fr/jcms/p_3325613/fr/decision-n-2022-0080/dc/sem-du-17-mars-2022-du-college-de-la-haute-autorite-de-sante-portant-autorisation-d-acces-precoce-de-la-specialite-lenvima
https://www.has-sante.fr/jcms/p_3328914/fr/decision-n-2022-0107/dc/sem-du-31-mars-2022-du-college-de-la-haute-autorite-de-sante-modifiant-la-decision-n-2022-0080/dc/sem-du-17-mars-2022-du-college-de-la-haute-autorite-de-sante-portant-autorisation-d-acces-precoce-de-la-specialite-lenvima
2022
false
false
false
France
Lenvatinib/Pembrolizumab Regimen
antineoplastic combined chemotherapy protocols
pembrolizumab
insurance, health, reimbursement
treatment outcome
endometrial neoplasms
Advanced Endometrial Carcinoma
neoplasm metastasis
neoplasm recurrence, local
Recurrent Endometrial Carcinoma
administration, oral
lenvatinib
protein kinase inhibitors
antineoplastic agents
evaluation of the transparency committee
lenvatinib

---
https://www.has-sante.fr/jcms/p_3321831/fr/kisplyx-lenvatinib-cancer-du-rein-uniquement-a-cellules-claires
2022
false
false
false
France
lenvatinib
protein kinase inhibitors
antineoplastic agents
treatment outcome
insurance, health, reimbursement
antineoplastic combined chemotherapy protocols
pembrolizumab
clear cell renal cell carcinoma
Lenvatinib/Pembrolizumab Regimen
Advanced Clear Cell Renal Cell Carcinoma
administration, oral
Product containing precisely lenvatinib (as lenvatinib mesilate) 10 milligram/1 each conventional release oral capsule (clinical drug)
Product containing precisely lenvatinib (as lenvatinib mesilate) 4 milligram/1 each conventional release oral capsule (clinical drug)
evaluation of the transparency committee
lenvatinib

---
https://www.has-sante.fr/jcms/p_3113418/fr/lenvima
2019
false
false
false
France
lenvatinib
treatment outcome
antineoplastic agents
protein kinase inhibitors
lenvatinib
adult
carcinoma, hepatocellular
administration, oral
evaluation of the transparency committee
Lenvima
phenylurea compounds
quinolines

---
https://www.has-sante.fr/portail/jcms/c_2834705/fr/kisplyx-lenvatinib-inhibiteur-de-tyrosine-kinase
https://www.has-sante.fr/portail/jcms/c_2834705/fr/kisplyx
2018
false
false
false
France
French
lenvatinib
treatment outcome
antineoplastic combined chemotherapy protocols
carcinoma, renal cell
adult
protein kinase inhibitors
protein kinase inhibitors
antineoplastic agents
antineoplastic agents
lenvatinib
administration, oral
protein-tyrosine kinases
receptor Protein-Tyrosine kinases
evaluation of the transparency committee
guidelines for drug use
insurance, health, reimbursement
disease-free survival
Everolimus
Tyrosine Kinase Inhibitors
lenvatinib
phenylurea compounds
quinolines
phenylurea compounds
quinolines

---
https://www.ema.europa.eu/medicines/human/EPAR/Kisplyx
2016
false
false
false
United Kingdom
French
English
syndication feed
summary of product characteristics
package leaflet
drug evaluation
lenvatinib
drug approval
europe
treatment outcome
drug interactions
antineoplastic combined chemotherapy protocols
carcinoma, renal cell
adult
protein kinase inhibitors
protein kinase inhibitors
antineoplastic agents
antineoplastic agents
lenvatinib
administration, oral
protein-tyrosine kinases
product surveillance, postmarketing
pregnancy
breast feeding
receptor Protein-Tyrosine kinases
drug evaluation, preclinical
Product containing precisely lenvatinib (as lenvatinib mesilate) 4 milligram/1 each conventional release oral capsule (clinical drug)
Product containing precisely lenvatinib (as lenvatinib mesilate) 10 milligram/1 each conventional release oral capsule (clinical drug)
Tyrosine Kinase Inhibitors
lenvatinib
phenylurea compounds
quinolines
phenylurea compounds
quinolines
phenylurea compounds
quinolines

---
https://hpr-rps.hres.ca/reg-content/sommaire-motif-decision-detailTwo.php?lang=fr&linkID=SBD00209
2016
false
false
false
Canada
French
English
summary of product characteristics
administration, oral
antineoplastic agents
antineoplastic agents
protein kinase inhibitors
protein kinase inhibitors
risk assessment
adult
thyroid neoplasms
Differentiated Thyroid Gland Carcinoma
Refractory Carcinoma
treatment outcome
Cancer Progression
drug approval
drug evaluation, preclinical
protein-tyrosine kinases
lenvatinib
canada
Lenvatinib Mesylate
Lenvatinib Mesylate
neoplasm recurrence, local
neoplasm metastasis
Tyrosine Kinase Inhibitors
lenvatinib
lenvatinib
phenylurea compounds
quinolines
phenylurea compounds
quinolines

---
Progrès thérapeutique mineur dans la prise en charge du cancer différencié de la thyroïde au stade localement avancé ou métastatique, réfractaire à l’iode radioactif
http://www.has-sante.fr/portail/jcms/c_2581320/fr/lenvima
http://www.has-sante.fr/portail/jcms/c_2581320/fr/lenvima-lenvatinib-inhibiteur-de-proteine-kinase
2015
false
false
false
France
French
administration, oral
antineoplastic agents
antineoplastic agents
protein kinase inhibitors
protein kinase inhibitors
risk assessment
adult
thyroid neoplasms
Differentiated Thyroid Gland Carcinoma
Refractory Carcinoma
treatment outcome
survival analysis
neoplasm metastasis
Locally Advanced Malignant Neoplasm
evaluation of the transparency committee
Cancer Progression
lenvatinib
guidelines for drug use
lenvatinib
lenvatinib
phenylurea compounds
quinolines
phenylurea compounds
quinolines

---
https://www.ema.europa.eu/medicines/human/EPAR/LENVIMA
2015
false
false
false
United Kingdom
French
English
package leaflet
summary of product characteristics
administration, oral
antineoplastic agents
antineoplastic agents
protein kinase inhibitors
protein kinase inhibitors
drug evaluation
risk assessment
adult
thyroid neoplasms
Differentiated Thyroid Gland Carcinoma
Refractory Carcinoma
treatment outcome
Cancer Progression
syndication feed
orphan drug production
drug approval
europe
drug interactions
pregnancy
breast feeding
drug evaluation, preclinical
continuity of patient care
product surveillance, postmarketing
protein-tyrosine kinases
lenvatinib
Tyrosine Kinase Inhibitors
lenvatinib
lenvatinib
phenylurea compounds
quinolines
phenylurea compounds
quinolines

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13/05/2024


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