Preferred Label : cholinesterase inhibitors;

MeSH definition : Drugs that inhibit cholinesterases. The neurotransmitter ACETYLCHOLINE is rapidly hydrolyzed, and thereby inactivated, by cholinesterases. When cholinesterases are inhibited, the action of endogenously released acetylcholine at cholinergic synapses is potentiated. Cholinesterase inhibitors are widely used clinically for their potentiation of cholinergic inputs to the gastrointestinal tract and urinary bladder, the eye, and skeletal muscles; they are also used for their effects on the heart and the central nervous system.;

MeSH synonym : anticholinesterases; drugs, anticholinesterase; anticholinesterase agents; anticholinesterase drugs; anti cholinesterases; inhibitors, cholinesterase; agents, anticholinesterase; anti-cholinesterases; Anticholinesterase Agent; Agent, Anticholinesterase; Anticholinesterase Drug; Drug, Anticholinesterase; Anticholinesterase; Anti-Cholinesterase; Anti Cholinesterase; Cholinesterase Inhibitor; Inhibitor, Cholinesterase;

MeSH hyponym : acetylcholinesterase inhibitors; cholinesterase inhibitors, irreversible; cholinesterase inhibitors, reversible; Inhibitors, Irreversible Cholinesterase; Irreversible Cholinesterase Inhibitors; Inhibitors, Reversible Cholinesterase; Reversible Cholinesterase Inhibitors; Inhibitors, Acetylcholinesterase; Acetylcholinesterase Inhibitor; Inhibitor, Acetylcholinesterase;

MeSH annotation : DF: CHOLINESTERASE INHIB;

Wikipedia link : https://en.wikipedia.org/wiki/Cholinesterase inhibitors;

Is substance : O;

action pharmacologique : O;

Details


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Drugs that inhibit cholinesterases. The neurotransmitter ACETYLCHOLINE is rapidly hydrolyzed, and thereby inactivated, by cholinesterases. When cholinesterases are inhibited, the action of endogenously released acetylcholine at cholinergic synapses is potentiated. Cholinesterase inhibitors are widely used clinically for their potentiation of cholinergic inputs to the gastrointestinal tract and urinary bladder, the eye, and skeletal muscles; they are also used for their effects on the heart and the central nervous system.

https://www.cbip.be/fr/articles/4528?folia=4520
2025
false
false
false
Belgium
French
journal article
pharmacovigilance note
drug interactions
anti-inflammatory agents, non-steroidal
cholinesterase inhibitors
risk
aged
peptic ulcer
alzheimer disease

---
https://dumas.ccsd.cnrs.fr/dumas-01492037
2017
false
true
false
France
French
dissertations, academic
cholinesterase inhibitors
residential facilities
memantine
alzheimer disease

---
https://www.has-sante.fr/portail/jcms/c_2679466/fr/medicaments-de-la-maladie-d-alzheimer-un-interet-medical-insuffisant-pour-justifier-leur-prise-en-charge-par-la-solidarite-nationale
2016
false
false
false
France
French
drug evaluation
alzheimer disease
treatment outcome
evaluation of the transparency committee
donepezil hydrochloride
donepezil
cholinesterase inhibitors
cholinesterase inhibitors
insurance, health, reimbursement
alzheimer disease
memantine
memantine
memantine hydrochloride
receptors, n-methyl-d-aspartate
excitatory amino acid antagonists
excitatory amino acid antagonists
administration, oral
administration, cutaneous
Rivastigmine
rivastigmine
galantamine
Galanthamine Hydrobromide
quality of life
galantamine
indans
piperidines
Donepezil

---
https://www.jle.com/fr/revues/gpn/e-docs/les_traitements_symptomatiques_dans_la_maladie_dalzheimer_en_2016_a_partir_des_centres_memoire_ressources_recherche_cmrr_en_france_308090/article.phtml
10.1684/pnv.2016.0629
2016
false
false
false
France
French
journal article
alzheimer disease
cholinesterase inhibitors
cholinesterase inhibitors
cholinesterase inhibitors
cholinesterase inhibitors
neurobehavioral manifestations
france

---
https://pharmacomedicale.org/medicaments/par-specialites/item/medicaments-de-la-plaque-neuromusculaire-les-points-essentiels
2016
false
false
false
France
French
drug information
cholinesterase inhibitors
neuromuscular blocking agents
botulinum antitoxin
drug, nos
myoneural junction
neuromuscular junction
essential
drugs, essential

---
https://pharmacomedicale.org/medicaments/par-specialites/item/stimulants-de-la-cognition-les-points-essentiels
2015
false
false
false
France
French
drug information
cognition disorders
excitatory amino acid antagonists
receptors, n-methyl-d-aspartate
cholinesterase inhibitors
cognition, nos
central nervous system stimulants
cognition
stimulator, nos
essential

---
http://www.cochrane.org/fr/CD001191/la-rivastigmine-pour-les-personnes-atteintes-de-la-maladie-dalzheimer
2015
false
false
false
France
United Kingdom
French
review of literature
treatment outcome
cholinesterase inhibitors
french abstract
Rivastigmine
Rivastigmine
alzheimer disease
cholinesterase inhibitors

---
http://www.cochrane.org/fr/CD006986
2014
false
false
false
United Kingdom
France
treatment outcome
review of literature
french abstract
myasthenia gravis
cholinesterase inhibitors

---
http://www.has-sante.fr/portail/jcms/c_1660673/fr/maladie-d-alzheimer-et-maladies-apparentees-diagnostic-et-prise-en-charge-de-l-apathie
http://www.has-sante.fr/portail/jcms/c_1766878/fr/apathie-argumentaire-scientifique
http://www.has-sante.fr/portail/jcms/c_1766877/fr/apathie-recommandations
2014
false
true
false
France
French
alzheimer disease
apathy
practice guideline
diagnosis, differential
prevalence
depressive disorder, major
caregivers
therapeutics
cholinesterase inhibitors
memantine
antidepressive agents

---
http://www.cochrane.org/fr/CD004746
2013
United Kingdom
France
French
meta-analysis
galantamine
cognition disorders
treatment outcome
dementia, vascular
cholinesterase inhibitors
nootropic agents
french abstract

---
http://www.cochrane.org/fr/CD007967
2012
false
true
false
United Kingdom
France
treatment outcome
review of literature
french abstract
cholinesterase inhibitors
schizophrenia

---
http://www.has-sante.fr/portail/jcms/c_1231960/place-des-medicaments-du-traitement-symptomatique-de-la-maladie-dalzheimer
http://www.has-sante.fr/portail/upload/docs/application/pdf/2012-03/questions_alzheimer_fiche_bum_mars_2012.pdf
2012
true
France
French
guidelines for drug use
practice guideline
Rivastigmine
donepezil
Galanthamine Hydrobromide
rivastigmine
galantamine
alzheimer disease
cholinesterase inhibitors
donepezil hydrochloride
nootropic agents
administration, oral
administration, cutaneous
transdermal patch
indans
piperidines
acetylcholinesterase
butyrylcholinesterase
drug evaluation
treatment outcome
Delayed-Action preparations
galantamine
excitatory amino acid antagonists
memantine
memantine hydrochloride
memantine
receptors, n-methyl-d-aspartate
evaluation of the transparency committee
Donepezil

---
http://www.cochrane.org/fr/CD009132
2012
United Kingdom
France
French
Cognitive Dysfunction
treatment outcome
meta-analysis
french abstract
cholinesterase inhibitors

---
https://www.jle.com/fr/revues/medecine/gpn/e-docs/00/04/74/B9/article.phtml
2012
France
French
Cardiotoxicity
cholinesterase inhibitors
review of literature
arrhythmias, cardiac

---
http://www.cochrane.org/fr/CD006504
http://www.cochrane.org/fr/CD006504/les-inhibiteurs-de-la-cholinesterase-sont-benefiques-pour-les-personnes-atteintes-de-la-maladie-de-parkinson-et-de-demence
2012
false
true
false
United Kingdom
France
treatment outcome
cognition disorders
meta-analysis
french abstract
cholinesterase inhibitors
lewy body disease
parkinson disease

---
https://www.boitedecision.ulaval.ca/boite-pdf/?tx_tmboites_tmboitesshow%5Bboite%5D=24&cHash=dc4d6155a20017ca6402459246b9200a
2012
false
false
false
false
Canada
French
decision making
popular works
cholinesterase inhibitors
alzheimer disease
scientific and technical information

---
http://www.cochrane.org/fr/CD005593
2012
United Kingdom
France
French
meta-analysis
cholinesterase inhibitors
alzheimer disease
treatment outcome
nootropic agents
french abstract

---
https://www.inspq.qc.ca/sites/default/files/publications/1199_medsystemenerveuxcanicules.pdf
2010
Canada
French
central nervous system agents
extreme heat
antidepressive agents
anticonvulsants
cholinesterase inhibitors
lithium
antipsychotic agents
antiparkinson agents
heat stroke
Drug-Related side effects and adverse reactions
guideline

---
http://www.john-libbey-eurotext.fr/fr/revues/medecine/nro/e-docs/00/04/4B/A8/resume.phtml
2009
false
France
French
Rivastigmine
alzheimer disease
cholinesterase inhibitors
piperidines
indans
galantamine
anticholinesterases
treatment outcome
memantine
excitatory amino acid antagonists
receptors, n-methyl-d-aspartate
memantine
journal article
Donepezil

---
http://www.has-sante.fr/portail/display.jsp?id=c_594386
http://www.has-sante.fr/portail/display.jsp?id=c_594403
2007
true
France
French
alzheimer disease
indans
piperidines
cholinesterase inhibitors
dopamine agents
galantamine
phenylcarbamates
memantine
excitatory amino acid antagonists
anti-dementia drugs
patient care management
guidelines for drug use

---
https://www.jle.com/fr/revues/medecine/med/e-docs/00/04/20/F6/resume.md?type=text.html
2006
France
French
alzheimer disease
continuity of patient care
cholinesterase inhibitors
social support
public assistance
institutionalization
journal article

---
https://minerva-ebp.be/fr/article/686
2006
false
false
minerva-ebm.be
Belgium
French
cholinesterase inhibitors
alzheimer disease
treatment outcome
critical appraisal or critical reading

---
https://minerva-ebp.be/fr/article/830
2005
false
false
minerva-ebm.be
Belgium
French
alzheimer disease
treatment outcome
memantine
excitatory amino acid antagonists
cholinesterase inhibitors
nootropic agents
drug therapy, combination
indans
piperidines
critical appraisal or critical reading
Donepezil

---
https://www.cadth.ca/fr/inhibiteurs-de-la-cholinesterase-pour-la-maladie-dalzheimer-examen-systematique-des-essais-cliniques
2005
true
Canada
French
Therapy cessation
alzheimer disease
cholinesterase inhibitors
Evidence-Based medicine
treatment outcome
canada
aged
disability evaluation
cholinesterase inhibitors
quality of life
alzheimer disease
prevalence
institutionalization
clinical trials as topic
indans
piperidines
galantamine
phenylcarbamates
data collection
anticholinesterases
meta-analysis
evaluation studies
technical report
french abstract
drug evaluation

---
https://minerva-ebp.be/fr/article/751
2005
false
false
minerva-ebm.be
Belgium
French
alzheimer disease
cholinesterase inhibitors
nootropic agents
treatment outcome
Cost-Benefit analysis
indans
piperidines
critical appraisal or critical reading
Donepezil

---
http://www.fmoq.org/Lists/FMOQDocumentLibrary/fr/Le%20M%C3%A9decin%20du%20Qu%C3%A9bec/Archives/2000%20-%202009/029infoPOEMs0503.pdf
2003
false
false
Canada
French
Sildenafil Citrate
Evidence-Based medicine
treatment outcome
cholinesterase inhibitors
alzheimer disease
irritable bowel syndrome
echinacea
plant preparations
common cold
antidepressive agents
erectile dysfunction
erectile dysfunction
hypertension
heart failure
blood pressure
risk factors
critical appraisal or critical reading

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24/05/2025


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