Preferred Label : Lenacapavir Sodium;
NCIt related terms : Sunlenca;
NCIt definition : The sodium salt form of lenacapavir, an inhibitor of human immunodeficiency virus
type 1 (HIV-1) capsid function, with activity against HIV. Upon administration, lenacapavir
targets and binds to the interface between HIV capsid protein (p24) subunits in hexamers.
This inhibits capsid function, including capsid-mediated nuclear uptake of preintegration
complexes, virion production and proper capsid core formation, thereby inhibiting
HIV-1 replication.;
UNII : BDT58WJ9WE;
CAS number : 2283356-12-5;
Drug name : Sunlenca;
NCI Metathesaurus CUI : CL1778580;
Origin ID : C186395;
UMLS CUI : C5670506;
Semantic type(s)
concept_is_in_subset
has_free_acid_or_base_form
is_salt_form_of
https://www.has-sante.fr/jcms/p_3392767/fr/sunlenca-lenacapavir-sodique-vih1-multiresistante-aux-medicaments
2022
false
false
false
France
French
evaluation of the transparency committee
treatment outcome
insurance, health, reimbursement
antiviral agents
Lenacapavir
Lenacapavir Sodium
injections, subcutaneous
administration, oral
lenacapavir
drug therapy, combination
adult
hiv infections
HIV-1
drug resistance, multiple, viral
multiresistant HIV-1 infection
---