NCIt synonyms : AR Degrader CC-94676; Androgen Receptor Degrader CC-94676;
NCIt definition : An orally bioavailable androgen receptor (AR) degrader, with potential antineoplastic
activity. Upon administration, gridegalutamide causes degradation of AR, prevents
AR-mediated signaling and inhibits the proliferation of AR-overexpressing tumor cells.
AR plays a key role in tumor cell proliferation in castration-resistant prostate cancer
(CRPC).;