Preferred Label : 4-OH-DiPT Prodrug RE104;
NCIt synonyms : 5-HT2A Agonist RE104; 5-Hydroxytryptamine Receptor 2A Agonist RE104;
NCIt definition : A prodrug form of the synthetic 5-hydroxytryptamine 2A receptor (5-HT2A) agonist 4-hydroxy-N,N-diisopropyltryptamine
(4-OH-DiPT), composed of a glutarate moiety linked to the phenolic functional group
of 4-OH-DiPT, with potential psychedelic activity. Upon administration of 4-OH-DiPT
prodrug RE104, the glutarate moiety is cleaved and the active moiety 4-OH-DiPT is
released. 4-OH-DiPT activates serotonin 2A (5-HT2A) receptors in the central nervous
system (CNS), mimicking the effects of serotonin, which may reduce depressive symptoms.;
Molecule name : RE 104; RE-104;
Origin ID : C217735;
concept_is_in_subset
- has_target
