Preferred Label : pentazocine;
MeSH definition : The first mixed agonist-antagonist analgesic to be marketed. It is an agonist at the
kappa and sigma opioid receptors and has a weak antagonist action at the mu receptor.
(From AMA Drug Evaluations Annual, 1991, p97);
CISMeF synonym : 17146-95-1 (Pentazocine lactate); 64024-15-3 (Pentazocine hydrochloride);
MeSH hyponym : Pentazocine Hydrochloride; talwin; Pentazocine Lactate; fortral; lexir; Lactate, Pentazocine; Hydrochloride, Pentazocine;
MeSH CAS label : 2,6-Methano-3-benzazocin-8-ol, 1,2,3,4,5,6-hexahydro-6,11-dimethyl-3-(3-methyl-2-butenyl)-,
(2alpha,6alpha,11R*)-;
MeSH Related Number : pentazocine lactate; pentazocine hydrochloride; 17146-95-1 (lactate); 359-83-1 (Pentazocine); 64024-15-3 (HCl); 1P2XIB510O; A36BXO4PPX;
Registry Number MeSH : 359-83-1;
Related CAS MeSH : 1P2XIB510O (Pentazocine lactate); A36BXO4PPX (Pentazocine hydrochloride);
Wikipedia link : https://en.wikipedia.org/wiki/Pentazocine;
Codes EINECS : 206-634-6;
Is substance : O;
UNII : RP4A60D26L;
InChIKey : VOKSWYLNZZRQPF-GDIGMMSISA-N;
Origin ID : D010423;
UMLS CUI : C0030873;
ATC code(s)
Allowable qualifiers
CISMeF manual mappings
Pharmacological action(s)
Record concept(s)
Related MeSH Supplementary Concept(s)
- JO 2871 [MeSH Supplementary Concept]
- KF 1820 [MeSH Supplementary Concept]
Semantic type(s)
UMLS correspondences (same concept)
Validated automatic mappings to BTNT
The first mixed agonist-antagonist analgesic to be marketed. It is an agonist at the
kappa and sigma opioid receptors and has a weak antagonist action at the mu receptor.
(From AMA Drug Evaluations Annual, 1991, p97)